DC26175NLX-101（F-15599）
F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist, with Ki of 3.4 nM.
View activity & pricesDC Chemicals · Research reagentsDC26175 
DC39022
DC12503
DC26111
DC31193
DC33443
DC10458
DC31161
DC22307
DC23413
DCAPI1471
DC11290
DC21710
DCAPI1439
DC24188
DC32105
DC43451
DCAPI1428
DC8771
DC26025
DC59005
DC60154
DC8607
DC39045
DC7079
DC60173
DC57073
DC8337
DC31745
DCAPI1072
DC10516
DC20250
DC23210
DC60059
DC11385
DCAPI1211
DC73953
DC32395
DC9772
DC65600
DC60493
DC20297
DC8441
DC36924
DCAPI1242
DCC0593
DC71430
DC26059
Other Research Tools
1099 products · Page 19 of 23
All small molecule research tools
DC26175DC39022BAY 2416964
BAY 2416964 is a 2-heteroaryl-3-oxo-2,3-dihydropyridazine-4-carboxamide compound and an aryl hydrocarbon receptor (AHR) antagonist extracted from patent WO2018146010A1, example 192, has an IC50 of 341 nM. AHR…
View activity & pricesDC12503STD1T
STD1T (USP2a inhibitor STD1T) is a hit-to-lead, small-molecule inhibitor of USP2a with IC50 of 3.3 uM in Ub-AMC assays, displays no activity against USP7 at 10 uM.
View activity & pricesDC26111Cevidoplenib
Cevidoplenib (SKI-O-703) is an orally available inhibitor of spleen tyrosine kinase (Syk), with potential anti-inflammatory and immunomodulating activities. Cevidoplenib is also the mesylate form of SKI-O-592.…
View activity & pricesDC31193Abiraterone Acetate (CB7630)
Abiraterone acetate is an FDA approved drug, and is an orally active acetate ester of the steroidal compound abiraterone with antiandrogen activity. Abiraterone acetate was approved by the U.S. Food and Drug…
View activity & pricesDC33443CCRIS 9056(Erucin)
Erucin is a sulforaphane analog and telomerase inhibitor found in cruciferous vegtables. It induces phase II enzyme activity, suppresses cellular proliferation in hepatocellular carcinoma cells, prevents 6-OHDA-induced…
View activity & pricesDC10458Delafloxacin（ABT-492）
Delafloxacin (RX-3341, ABT-492) is a fluoroquinolone antibiotic agent.
View activity & pricesDC31161AP24534 hydrochloride
Ponatinib, also known as AP24534 is an oral drug for the treatment of chronic myeloid leukemia (CML) and Philadelphia chromosome–positive (Ph+) acute lymphoblastic leukemia (ALL). It is a multi-targeted tyrosine-kinase…
View activity & pricesDC22307DMX-5804
DMX-5804 is a potent, orally active and selective MAP4K4 inhibitor, with an IC50 of 3 nM, a pIC50 of 8.55 for human MAP4K4, less potent on MINK1/MAP4K6 (pIC50, 8.18), and TNIK/MAP4K7 (pIC50, 7.96). DMX-5804 enhances…
View activity & pricesDC23413BTRX335140
BTRX-335140 (CYM-53093) is a potent and selective, orally active κ opioid receptor (KOR) antagonist, has antagonist activity for κOR, μOR and δOR with IC50 values of 0.8 nM, 110 nM, and 6500 nM,…
View activity & pricesDCAPI1471Arabinofuranosylcytosine
For the detailed information of Arabinofuranosylcytosine, the solubility of Arabinofuranosylcytosine in water, the solubility of Arabinofuranosylcytosine in DMSO, the solubility of Arabinofuranosylcytosine in PBS…
View activity & pricesDC11290QC-3611
QC-3611 is a selective inhibitor of JARID1A/1B, which is a target existing in various tumors (JARID1A IC50 = 13 nM ;JARID1B IC50 = 2 nM). QC-3611 is promisingly to be used as an antineoplastic drug.
View activity & pricesDC21710SU-909
SU-909 (SU909, IKKα-IN-48) is a potent, selective IKKα inhibitor with Ki of 0.08±0.07 uM, 10-20-fold selectivity over IKKβ (IC50=1.0±0.28 uM); inhibits FCS-stimulated phosphorylation of p100 in U2OS cells with IC50 of…
View activity & pricesDCAPI1439Ropivacaine HCL
Ropivacaine HCl is an anaesthetic agent and blocks impulse conduction in nerve fibres through inhibiting sodium ion influx reversibly.Ropivacaine is a new long-acting local anesthetic, with vasoconstrictive properties.…
View activity & pricesDC24188Trenbolone acetate
Trenbolone acetate (RU-1697,17beta-TBOH) is a potent testosterone analog and selective androgen receptor modulator, is an androgen ester and a long-acting prodrug of trenbolone; shows SARM-like effects as it binds to…
View activity & pricesDC32105Ganaxolone
Ganaxolone, also known as CCD 1042 and C1042, is a CNS-selective GABAA modulator that acts on well-characterized targets in the brain known to have anxiolytic and anticonvulsant effects. Ganaxolone protects against…
View activity & pricesDC434514BP-TQS
Potent Allosteric Agonist-Positive Allosteric Modulator of α7 Nicotinic Acetylcholine Receptors
View activity & pricesDCAPI1428Clofarabine
Clofarabine(Clolar; Clofarex) inhibits the enzymatic activities of ribonucleotide reductase (IC50 = 65 nM) and DNA polymerase.
View activity & pricesDC8771Tucatinib (Irbinitinib,ARRY-380)
Tucatinib (Irbinitinib; ARRY-380; ONT-380) is a potent and selective HER2 inhibitor with an IC50 of 8 nM.
View activity & pricesDC26025INCB086550(INCB-086550)
INCB086550 is an orally available, small molecule inhibitor of PD-L1 with potential immune checkpoint inhibitory and antineoplastic activities. In vitro, INCB086550 selectively and potently blocked the PD-L1/PD-1…
View activity & pricesDC59005Ozanimod hydrochloride
Ozanimod is a potent and selective S1P1 and S1P5 receptor agonist with EC50s of 410±160 pM and 11±4.3 nM in 35S-GTPγS binding, respectively.
View activity & pricesDC60154Miclxin
Miclxin, a Novel MIC60 Inhibitor, Induces Apoptosis via Mitochondrial Stress in β-Catenin Mutant Tumor Cells
View activity & pricesDC8607Tideglusib(NP-031112)
Tideglusib is an irreversible GSK-3 inhibitor with IC50s of 5 nM and 60 nM for GSK-3βWT (1 h preincubation) and GSK-3βC199A (1 h preincubation), respectively.
View activity & pricesDC39045Apostatin-1 (Apt-1)
Apostatin-1 (Apt-1) is a novel TRADD inhibitor.Apostatin-1 inhibits RIPK1-dependent apoptosis (RDA) with IC50 of 1.28 μM and shows no significant off-target activity on 97 kinases in KINOME scan profiling.Inhibition of…
View activity & pricesDC7079Alvelestat (AZD9668)
Alvelestat (AZD9668) is a novel, oral inhibitor of neutrophil elastase (NE) with the pIC50 of 7.9 for Human NE.
View activity & pricesDC60173BR-103354
BR103354 is a novel fibroblast activation protein (FAP) inhibitor with anti-diabetic and anti-steatotic effects.
View activity & pricesDC57073VX-150
VX-150 is an orally active, highly selective NaV1.8 inhibitor. VX-150 has the potential for various pain indications research[1].
View activity & pricesDC8337Fluensulfone
Fluensulfone is a new nematicide for chemical control of plant parasitic nematodes.
View activity & pricesDC31745Methacholine Chloride
Methacholine chloride is used to constrict airway smooth muscle and to assess bronchial reactivity. Methacholine chloride is a cholinergic agonist and parasympathomimetic bronchoconstrictor. A metabolically stable…
View activity & pricesDCAPI1072Diphenhydramine HCl (Benadryl)
For the detailed information of Diphenhydramine HCl (Benadryl), the solubility of Diphenhydramine HCl (Benadryl) in water, the solubility of Diphenhydramine HCl (Benadryl) in DMSO, the solubility of Diphenhydramine HCl…
View activity & pricesDC10516LW6(CAY10585)
LW6 is a novel HIF-1 inhibitor with an IC50 of 4.4 μM.
View activity & pricesDC20250NRX2663
NRX-2663 is an enhancer of the interaction between β-catenin, and its cognate E3 ligase, SCFβ-TrCP. NRX-2663 enhances the binding of β-catenin peptide for β-TrCP with an EC50 of 22.9 µM and a Kd of 54.8 nM1.
View activity & pricesDC23210SZL P1-41
SZL P1-41 is Skp2 inhibitor, selectively suppresses Skp2 E3 ligase activity, but not activity of other SCF complexes.
View activity & pricesDC60059Capmatinib hydrochloride
Capmatinib, also known as INCB28060 and INC280, is an orally bioavailable inhibitor of the proto-oncogene c-Met with potential antineoplastic activity. c-Met inhibitor INC280 selectively binds to c-Met, thereby…
View activity & pricesDC11385Trofinetide(NNZ2566)
Trofinetide, a synthetic analogue of the endogenous N-terminus tripeptide, Glycine-Proline-Glutamate (GPE), has been shown to be neuroprotective in animal models of brain injury.
View activity & pricesDCAPI1211L-Thyroxine
For the detailed information of L-Thyroxine, the solubility of L-Thyroxine in water, the solubility of L-Thyroxine in DMSO, the solubility of L-Thyroxine in PBS buffer, the animal experiment（test） (test) of…
View activity & pricesDC73953CPAG-1
CPAG-1 (PGRMC2 activator CPAG-1) is a small-molecule activator of PGRMC2. CPAG-1 treatment had no effect on weight or food intake but treated mice had reduced fasting glycemia and insulin levels. CPAG-1 decreased…
View activity & pricesDC32395Niraparib tosylate hydrate
Niraparib, also know as MK-4827, is an inhibitor of poly (ADP-ribose) polymerase (PARP) with potential antineoplastic activity.
View activity & pricesDC9772Efinaconazole(KP-103)
Efinaconazole(KP-103) is a novel triazole antifungal drug currently under development as a topical treatment for onychomycosis.
View activity & pricesDC6560042-(2-Tetrazolyl)rapamycin
42-(2-Tetrazolyl)rapamycin is a prodrug compound of a rapamycin analog extracted from patent US 20080171763 A1, Example 1. Rapamycin is a specific mTOR inhibitor.
View activity & pricesDC60493BEBT-809
BEBT-809 is a GPR75 antagonist for rat CYP4F2 and CYP4A11 with IC50 of and 15.76 nM and 33.16 nM, respectively.
View activity & pricesDC202976-Hydroxy-DL-DOPA
6-Hydroxy-DOPA is a selective and effective allosteric inhibitor of the RAD52 ssDNA binding domain. 6-Hydroxy-DOPA can be used for the research of cancer[1].
View activity & pricesDC8441Nitenpyram
For the detailed information of Nitenpyram, the solubility of Nitenpyram in water, the solubility of Nitenpyram in DMSO, the solubility of Nitenpyram in PBS buffer, the animal experiment (test) of Nitenpyram, the cell…
View activity & pricesDC36924NNMTi
NNMTi is a potent nicotinamide N-methyltransferase (NNMT) inhibitor (IC50=1.2 μM) and selectively binds to the NNMT substrate-binding site residues[1]. NNMTi promotes myoblast differentiation in vitro and enhances…
View activity & pricesDCAPI1242Isoniazid(Tubizid)
Isoniazid is an antibacterial agent used primarily as a tuberculostatic.Target: AntibacterialIsoniazid is a prodrug and must be activated by a bacterial catalase-peroxidase enzyme that in M. tuberculosis is called KatG…
View activity & pricesDCC0593Sotorasib racemate
Sotorasib racemate (Compound A) is an orally active racemate of Sotorasib, a covalent inhibitor of KRAS G12C mutant which induces adaptive feedback activation of MAPK pathway. Sotorasib racemate also exerts inhibitor…
View activity & pricesDC71430NHS-NH-(diethylamino)ethyl benzoate
NHS-NH-(diethylamino)ethyl benzoate is a compound that can be used for N-glycan labeling.
View activity & pricesDC26059Diprotin A
Diprotin A is a tripeptide inhibitor of dipeptidyl peptidase 4 (DPP-4; IC50 = 1.1 μg/ml).It inhibits degradation of glucagon-like peptide 1 in culture with insulin-secreting BRIN-BD11 rat pancreatic β-cells when used…
View activity & prices