STD1T chemical structure
Chemical structureResearch use only
CAT. NO. DC12503Featured

STD1T

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TotalUS$750
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Product overview

Description & Application

STD1T (USP2a inhibitor STD1T) is a hit-to-lead, small-molecule inhibitor of USP2a with IC50 of 3.3 uM in Ub-AMC assays, displays no activity against USP7 at 10 uM.

ParameterValue
Chemical Name2-(2-((5-(thiophen-2-yl)isoxazol-3-yl)methoxy)acetamido)-4,5,6,7-tetrahydrobenzo[b]thiophene-3-carboxamide
CAS No.893075-58-6
SynonymsUSP2a inhibitor STD1T
FormulaC19H19N3O4S2
M.Wt417.498
SMILESC12CCCCC=1C(C(N)=O)=C(NC(=O)COCC1C=C(C3SC=CC=3)ON=1)S2
Purity>98%
Storage2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Biological Activity

STD1T (USP2a inhibitor STD1T) is a hit-to-lead, small-molecule inhibitor of USP2a with IC50 of 3.3 uM in Ub-AMC assays, displays no activity against USP7 at 10 uM.

In Vitro

No in vitro data are provided in the current product source. Contact us for further information.

In Vivo

No in vivo data are provided in the current product source. Contact us for further information.

References & source

1. Tomala MD, et al. Eur J Med Chem. 2018 Apr 25;150:261-267.

DC Chemicals original product information

Published experimental findings depend on the model and assay conditions. They do not guarantee equivalent performance in every application. For laboratory research use only.

Product documentation

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Handling guide

2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

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