PPAR

13 products · Page 1 of 1

All small molecule research tools

DC10700

Seladelpar

Seladelpar is an orally active, potent (50% effect concentration EC50 2 nM), and specific PPAR-δ agonist.

View activity & prices

DC1035

GSK3787

GSK3787 is a selective and irreversible peroxisome proliferator-activated receptor δ (PPARδ) antagonist with pIC50 of 6.6.

View activity & prices

DC1036

GSK-0660

GSK0660 is a potent antagonist of PPARβ and PPARδ, with IC50s of 155 nM for both isoforms.

View activity & prices

DC4233

GW501516

GW 501516 is a PPARδ agonist with an EC50 of 1.1 nM.

View activity & prices

DC1034

WY14643 (Pirinixic Acid)

Pirinixic acid (Wy-14643) is a potent agonist of PPARα, with EC50s of 0.63 μM, 32 μM for murine PPARα and PPARγ, and 5.0 μM, 60 μM, 35 μM for human PPARα, PPARγ and PPARδ, respectively.

View activity & prices

DC11360

Pemafibrate

Pemafibrate is a potent PPARα agonist, with EC50s of 1 nM, 1.10 μM and 1.58 μM for h-PPARα, h-PPARγ and h-PPARδ, respectively, and possesses lipid-lowering effect.

View activity & prices

DC7412

R(+)-Etomoxir (sodium salt)

(R)-Etomoxir sodium salt is the R-form of Etomoxir sodium salt, acts as an inhibitorof carnitine palmitoyltransferase I (CPT-I), and inhibits palmitate β-oxidation in human, rat and guinea pig.

View activity & prices

DC9904

GW0742

GW0742 is a high affinity PPAR β/δ agonist with an IC50 of 1 nM for human PPARδ, and EC50s of 1 nM, 1.1 μM and 2 μM for human PPARδ, PPARα, and PPARγ, respectively.

View activity & prices

DC9602

Balaglitazone

Balaglitazone is a selective partial PPARγ agonist with an EC50 of 1.351 μM for human PPARγ.

View activity & prices

DC9601

T0070907

T0070907 is a potent PPARγ antagonist with a Ki of 1 nM.

View activity & prices

DC9252

BMS-687453

BMS-687453 is a potent and selective PPARα agonist, with an EC50 and IC50 of 10 nM and 260 nM for human PPARα and 4100 nM and >15000 nM for PPARγ in PPAR-GAL4 transactivation assays.

View activity & prices

DCAPI1413

pioglitazone hydrochloride

For the detailed information of pioglitazone hydrochloride, the solubility of pioglitazone hydrochloride in water, the solubility of pioglitazone hydrochloride in DMSO, the solubility of pioglitazone hydrochloride in…

View activity & prices

DC2079

GW-9662

GW9662 is a potent and selective PPARγ antagonist with an IC50 of 3.3 nM, showing 10 and 1000-fold selectivity over PPARα and PPARδ, respectively.

View activity & prices