Chemical structureResearch use only

CAT. NO. DC60874Featured

SKPer1 (XMU-MP-8)

Name: SKPer1 (XMU-MP-8)
Brand: DC Chemicals
SKU: DC60874
Price: 500.0 USD

Pack Sizes & Prices

TotalUS$500

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Product overview

Description & Application

SKPer1 (XMU-MP-8) is a small-molecule degrader of SKP2 that triggers degradation of the oncoprotein SKP2 and specifically kills SKP2-expressing cancer cells.

Parameter	Value
Chemical Name	SKPer1 (XMU-MP-8)
Formula	C26H21F3N8S
M.Wt	534.57
SMILES	CN1N=CC2=C1N=C(C1=CC(NC(=S)NC3=CC=CC(C(F)(F)F)=C3)=CC=C1)N=C2NCC1=CC=CN=C1
Purity	98%
Storage	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Biological Activity

SKPer1 (XMU-MP-8) is a small-molecule degrader of SKP2 that triggers degradation of the oncoprotein SKP2 and specifically kills SKP2-expressing cancer cells.

In Vitro

No in vitro data are provided in the current product source. Contact us for further information.

In Vivo

No in vivo data are provided in the current product source. Contact us for further information.

References & source

DC Chemicals original product information

Published experimental findings depend on the model and assay conditions. They do not guarantee equivalent performance in every application. For laboratory research use only.

Product documentation

View online datasheet Request COA / MSDS

Refer to the certificate supplied with your lot for batch-specific release results.

Handling guide

2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Solution calculator

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