DC10832(E/Z)-4-hydroxy Tamoxifen
(E/Z)-4-Hydroxytamoxifen is a racemic compound of (Z)-4-Hydroxytamoxifen and (E)-4-Hydroxytamoxifen isomers. (E/Z)-4-Hydroxytamoxifen is an estrogen receptor modulator.
View activity & pricesDC Chemicals · Research reagentsDC10832 
DC8922
DC9268
DC40118
DC7372
DC8265
DC44905
DC70851
DC10846
DC7735
DCAPI1501
DC10182
DC10077
Estrogen Receptor/ERR
13 products · Page 1 of 1
All small molecule research tools
DC10832DC8922Bazedoxifene
Bazedoxifene is a selective estrogen receptor modulator (SERM) currently in development for osteoporosis prevention and treatment.modulatorPreclinical and clinical studies with bazedoxifene demonstrate more tissue…
View activity & pricesDC9268AZD9496
AZD9496 is a potent and selective estrogen receptor (ERα) antagonist with an IC50 of 0.28 nM.
View activity & pricesDC40118Giredestrant
Giredestrant (GDC-9545), a non-steroidal ER ligand, is an orally active and selective estrogen receptor (ER) antagonist. Giredestrant potently competes with estradiol for binding and induces a conformational change…
View activity & pricesDC7372Bazedoxifene-Acetate
Bazedoxifene acetate is a third generation selective estrogen receptor modulator (SERM) with IC50s of 26 and 99 nM for ERα and ERβ, respectively.
View activity & pricesDC8265Endoxifen
Endoxifen Z-isomer is the most important Tamoxifen metabolite responsible for eliciting the anti-estrogenic effects of this drug in breast cancer cells expressing estrogen receptor-alpha (ERα). Endoxifen inhibits hERG…
View activity & pricesDC44905Vepdegestrant (ARV-471)
ARV-471 is a best-in-class, orally active estrogen receptor (ER) PROTAC degrader. ARV-471 is developed for the research of breast cancer.
View activity & pricesDC70851TTC-352
TTC-352 is a synthetic selective estrogen mimic acts as estrogen receptor (ER) partial agonist for the treatment of endocrine-resistant breast cancer.TTC-352 yields an H-bond with Glu353, allows Asp351-to-helix 12…
View activity & pricesDC10846PHTPP
PHTPP is a selective ERβ antagonist.
View activity & pricesDC7735XCT790
XCT-790 is a potent, selective and inverse agonist of estrogen-related receptor alpha(ERRα); induces cell death in chemotherapeutic resistant cancer cells.XCT-790 induced cell death in HepG2 hepatocarcinoma and its…
View activity & pricesDCAPI1501Lasofoxifene tartrate
Lasofoxifene Tartrate is a non-steroidal selective estrogen receptor modulator (SERM).
View activity & pricesDC10182Elacestrant (dihydrochloride)
Elacestrant dihydrochloride (RAD1901 dihydrochloride) is a selective and orally available estrogen receptor (ERR) degrader with IC50 values of 48 and 870 nM for ERα and ERβ, respectively.
View activity & pricesDC10077WAY-200070
WAY-200070 is a selective estrogen receptor β (ERRβ) agonist with an IC50 of 2.3 nM.
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