Chemical structureResearch use only

CAT. NO. DC70046Featured

MRTX 0902

Name: MRTX 0902
Brand: DC Chemicals
SKU: DC70046
Price: 900.0 USD

Pack Sizes & Prices

TotalUS$900

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Product overview

Description & Application

MRTX0902 is a potent SOS1 inhibitor with an IC50 of 46 nM (WO2021127429A1; Example 12-10).

Parameter	Value
Chemical Name	MRTX 0902
CAS No.	2654743-22-1
Synonyms	MRTX0902
Formula	C22H24N6O
M.Wt	388.475
SMILES	N#CC1=CC=CC([C@H](NC2=NN=C(C)C3=CN=C(N4CCOCC4)C=C32)C)=C1C
Purity	>98%
Storage	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Biological Activity

MRTX0902 is a potent SOS1 inhibitor with an IC50 of 46 nM (WO2021127429A1; Example 12-10).

In Vitro

No in vitro data are provided in the current product source. Contact us for further information.

In Vivo

No in vivo data are provided in the current product source. Contact us for further information.

References & source

[1]. Matthew Arnold Marx, et al. Sos1 inhibitors. WO2021127429A1.

[2]. Matthew Arnold Marx, et al. Sos1 inhibitors. WO2021127429A1.

DC Chemicals original product information

Published experimental findings depend on the model and assay conditions. They do not guarantee equivalent performance in every application. For laboratory research use only.

Product documentation

View online datasheet Request COA / MSDS

Refer to the certificate supplied with your lot for batch-specific release results.

Handling guide

2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Solution calculator

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