DC Chemicals · Product datasheet

MRTX 0902 — Datasheet

CAT. NO. DC70046

Product page and current package options

ParameterValue
Chemical NameMRTX 0902
CAS No.2654743-22-1
SynonymsMRTX0902
FormulaC22H24N6O
M.Wt388.475
SMILESN#CC1=CC=CC([C@H](NC2=NN=C(C)C3=CN=C(N4CCOCC4)C=C32)C)=C1C
Purity>98%
Storage2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Biological Activity

MRTX0902 is a potent SOS1 inhibitor with an IC50 of 46 nM (WO2021127429A1; Example 12-10).

In Vitro

No in vitro data are provided in the current product source. Contact us for further information.

In Vivo

No in vivo data are provided in the current product source. Contact us for further information.

References & source

[1]. Matthew Arnold Marx, et al. Sos1 inhibitors. WO2021127429A1.

[2]. Matthew Arnold Marx, et al. Sos1 inhibitors. WO2021127429A1.

DC Chemicals original product information

Published experimental findings depend on the model and assay conditions. They do not guarantee equivalent performance in every application. For laboratory research use only.

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