Cilofexor is a farnesoid X receptor (FXR) agonist.
| Parameter | Value |
|---|---|
| Chemical Name | Cilofexor |
| CAS No. | 1418274-28-8 |
| Synonyms | Cilofexor;PX104;YUN2306954;GS 9674;2-(3-(2-chloro-4-((5-cyclopropyl-3-(2,6-dichlorophenyl)isoxazol-4-yl)methoxy)phenyl)-3-hydroxyazetidin-1-yl)isonicotinic acid;2-[3-[2-chloro-4-[[5-cyclopropyl-3-(2,6-dichlorophenyl)-1,2-oxazol-4-yl]methoxy]phenyl]-3-hydroxyazetidin-1-yl]pyridine-4-carboxylic acid;Cilofexor [INN];Cilofexor (GS(c)\\9674);GTPL10644;BCP29283;BDBM50511109;GS9674;s6547;DB15168;example 13/9 [US1 |
| Formula | C28H22Cl3N3O5 |
| M.Wt | 586.8504 |
| SMILES | ClC1C([H])=C(C([H])=C([H])C=1C1(C([H])([H])N(C2C([H])=C(C(=O)O[H])C([H])=C([H])N=2)C1([H])[H])O[H])OC([H])([H])C1C(C2C(=C([H])C([H])=C([H])C=2Cl)Cl)=NOC=1C1([H])C([H])([H])C1([H])[H] |
| Purity | >98% |
| Storage | 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO |
Cilofexor is a farnesoid X receptor (FXR) agonist.
No in vitro data are provided in the current product source. Contact us for further information.
No in vivo data are provided in the current product source. Contact us for further information.
Published experimental findings depend on the model and assay conditions. They do not guarantee equivalent performance in every application. For laboratory research use only.
Refer to the certificate supplied with your lot for batch-specific release results.
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