Trpm2 Inhibitor A23 chemical structure
Chemical structureResearch use only
CAT. NO. DCC5248Featured

Trpm2 Inhibitor A23

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Product overview

Description & Application

Novel selective inhibitor of the transient receptor potential melastatin 2 (TRPM2) channel, exhibiting TRPM2 selectivity over TRPM8 and TRPV1 channels as well as phospholipase A2 and showing neuroprotective activity in vitro, and significantly reducing ce

ParameterValue
Chemical NameTrpm2 Inhibitor A23
CAS No.2765256-12-8
SynonymsTrpm2-Inhibitor-A23
FormulaC23H16F3NO3
M.Wt411.38
SMILESO=C(/C=C/C1=CC=C(C2=CC(C(F)(F)F)=CC=C2)C=C1)NC1=C(C(=O)O)C=CC=C1
Purity>98%
Storage2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Biological Activity

Novel selective inhibitor of the transient receptor potential melastatin 2 (TRPM2) channel, exhibiting TRPM2 selectivity over TRPM8 and TRPV1 channels as well as phospholipase A2 and showing neuroprotective activity in vitro, and significantly reducing ce

In Vitro

No in vitro data are provided in the current product source. Contact us for further information.

In Vivo

No in vivo data are provided in the current product source. Contact us for further information.

References & source

DC Chemicals original product information

Published experimental findings depend on the model and assay conditions. They do not guarantee equivalent performance in every application. For laboratory research use only.

Product documentation

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Handling guide

2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

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