amyloid P-IN-1(GSK3039294) chemical structure
Chemical structureResearch use only
CAT. NO. DC9717Featured

amyloid P-IN-1(GSK3039294)

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TotalUS$700
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Product overview

Description & Application

pharmaceutical compositions comprising the same and the use of the same for treatment of diseases or disorders wherein depletion of serum amyloid P component (SAP) would be beneficial, including amyloidosis, Alzheimer's disease, type 2 diabetes mellitus and osteoarthritis.

ParameterValue
CAS No.1819986-22-5
SynonymsGSK3039294;GSK-3039294;GSK 3039294
FormulaC30H44N2O14
M.Wt656.68
SMILESC1(CCOCC1)OC(=O)OCOC([C@H]1N(C(=O)CCCCC(=O)N2CCC[C@H]2C(=O)OCOC(=O)OC2CCOCC2)CCC1)=O
Purity>98%
Storage2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Biological Activity

pharmaceutical compositions comprising the same and the use of the same for treatment of diseases or disorders wherein depletion of serum amyloid P component (SAP) would be beneficial, including amyloidosis, Alzheimer's disease, type 2 diabetes mellitus and osteoarthritis.

In Vitro

No in vitro data are provided in the current product source. Contact us for further information.

In Vivo

No in vivo data are provided in the current product source. Contact us for further information.

References & source

[1]. PCT Int. Appl. (2015), WO 2015165833 A1 20151105.

[2]. U.S. Pat. Appl. Publ. (2016), US 20160081983 A1 20160324.

DC Chemicals original product information

Published experimental findings depend on the model and assay conditions. They do not guarantee equivalent performance in every application. For laboratory research use only.

Product documentation

Refer to the certificate supplied with your lot for batch-specific release results.

Handling guide

2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

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