NUCC-0200590 chemical structure
Chemical structureResearch use only
CAT. NO. DC73618Featured

NUCC-0200590

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TotalUS$450
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Product overview

Description & Application

NUCC-0200590 is a small-molecule inhibitor of the TRIP8b-HCN interaction with IC50 of 7.0 uM in AlphaScreen assays, effectively disrupts the TRIP8b-HCN interaction in vitro and in vivo.

ParameterValue
Chemical NameNUCC-0200590
CAS No.1060461-67-7
SynonymsNUCC0200590,NUCC 0200590
FormulaC27H29ClFN3O2
M.Wt482
SMILESCN1CCN(CC2=CC(C3=CC=C(F)C=C3)=CC=C2OCC(=O)NCC2=CC=C(Cl)C=C2)CC1
Purity98%

Biological Activity

NUCC-0200590 is a small-molecule inhibitor of the TRIP8b-HCN interaction with IC50 of 7.0 uM in AlphaScreen assays, effectively disrupts the TRIP8b-HCN interaction in vitro and in vivo.

In Vitro

No in vitro data are provided in the current product source. Contact us for further information.

In Vivo

No in vivo data are provided in the current product source. Contact us for further information.

References & source

DC Chemicals original product information

Published experimental findings depend on the model and assay conditions. They do not guarantee equivalent performance in every application. For laboratory research use only.

Product documentation

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