VU0606170 chemical structure
Chemical structureResearch use only
CAT. NO. DC70890Featured

VU0606170

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Product overview

Description & Application

VU 0606170 (also referred to as VU0606170) is a selective inhibitor of the sodium-activated potassium channel KNa1.1, also known as Slack or Slo2.2. This compound has shown specificity for Slack channels over other related potassium channels, making it a valuable tool for studying the physiological and pathological roles of KNa1.1.

ParameterValue
Chemical NameN-(5-chloro-2-methoxyphenyl)-2-{4-(4-methylpiperidin-1-yl)sulfonylpiperazin-1-yl}acetamide
CAS No.879054-55-4
SynonymsN-(5-chloro-2-methoxyphenyl)-2-{4-(4-methylpiperidin-1-yl)sulfonylpiperazin-1-yl}acetamide;VU0606170-1;N-(5-Chloro-2-methoxy-phenyl)-2-[4-(4-methyl-piperidine-1-sulfonyl)-piperazin-1-yl]-acetamide;N-(5-chloro-2-methoxyphenyl)-2-[4-(4-methylpiperidin-1-yl)sulfonylpiperazin-1-yl]acetamide;VU0606170;GLXC-26400;F3230-0289;CHEMBL1730394;SMR000606669;BRD-K98364914-001-07-8;BDBM50607064;N-(5-chloro-2-methoxyphenyl)-2-(4-((4-methylpiperidin-1-yl)sulfonyl)piperazin-1-yl)acetamide;AKOS000747558;879054-55-4;HMS2913A08;MLS001222086
FormulaC19H29ClN4O4S
M.Wt444.975962400436
SMILESClC1C=CC(=C(C=1)NC(CN1CCN(CC1)S(N1CCC(C)CC1)(=O)=O)=O)OC
Purity>98%
Storage2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Biological Activity

VU 0606170 (also referred to as VU0606170) is a selective inhibitor of the sodium-activated potassium channel KNa1.1, also known as Slack or Slo2.2. This compound has shown specificity for Slack channels over other related potassium channels, making it a valuable tool for studying the physiological and pathological roles of KNa1.1.

In Vitro

No in vitro data are provided in the current product source. Contact us for further information.

In Vivo

No in vivo data are provided in the current product source. Contact us for further information.

References & source

DC Chemicals original product information

Published experimental findings depend on the model and assay conditions. They do not guarantee equivalent performance in every application. For laboratory research use only.

Product documentation

Refer to the certificate supplied with your lot for batch-specific release results.

Handling guide

2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

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