Chemical structureResearch use only

CAT. NO. DC6312Featured

SB525334

Name: SB525334
Brand: DC Chemicals
SKU: DC6312
Price: 350.0 USD

Pack Sizes & Prices

TotalUS$350

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Product overview

Description & Application

SB 525334 is a potent and selective transforming growth factor β1 receptor (ALK5) inhibitor with an IC50 of 14.3 nM.

Parameter	Value
Chemical Name	6-(2-tert-butyl-4-(6-methylpyridin-2-yl)-1H-imidazol-5-yl)quinoxaline
CAS No.	356559-20-1
Synonyms	SB-525334,SB 525334
Formula	C21H21N5
M.Wt	343.42
SMILES	N1C2C(=CC(C3NC(C(C)(C)C)=NC=3C3=NC(C)=CC=C3)=CC=2)N=CC=1
Purity	99%
Storage	2 years -20°C powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Biological Activity

SB 525334 is a potent and selective transforming growth factor β1 receptor (ALK5) inhibitor with an IC50 of 14.3 nM.

In Vitro

No in vitro data are provided in the current product source. Contact us for further information.

In Vivo

No in vivo data are provided in the current product source. Contact us for further information.

References & source

DC Chemicals original product information

Published experimental findings depend on the model and assay conditions. They do not guarantee equivalent performance in every application. For laboratory research use only.

Product documentation

View online datasheet Request COA / MSDS

Refer to the certificate supplied with your lot for batch-specific release results.

Handling guide

2 years -20°C powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Solution calculator

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