Trotabresib (CC-90010) chemical structure
Chemical structureResearch use only
CAT. NO. DC41049Featured

Trotabresib (CC-90010)

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Product overview

Description & Application

CC-90010 (compound 1) is a reversible and orally active BET inhibitor. CC-90010 is applied in the study for advanced solid tumors

ParameterValue
Chemical NameUnii-K424WH3WU0
CAS No.1706738-98-8
SynonymsK424WH3WU0;Trotabresib;Trotabresib [USAN];BDBM285044;US10023592, Example 89;QC5487;WHO 11839;Cn1cc(-c2cc(ccc2OCC2CC2)S(C)(=O)=O)c2ccccc2c1=O;4-[2-(cyclopropylmethoxy)-5-methylsulfonylphenyl]-2-methylisoquinolin-1-one;1(2H)-Isoquinolinone, 4-(2-(cyclopropylmethoxy)-5-(methylsulfonyl)phenyl)-2-methyl-;4-(2-(cyclopropylmethoxy)-5-(methylsulfonyl)phenyl)-2-methylisoquinolin-1(2H)-one;4-[2-(cyclopropylmethoxy)- 5-methylsulfonylphenyl]-2- ;Unii-K424WH3WU0;CC-90010
FormulaC21H21NO4S
M.Wt383.4607
SMILESS(C([H])([H])[H])(C1C([H])=C([H])C(=C(C=1[H])C1=C([H])N(C([H])([H])[H])C(C2=C([H])C([H])=C([H])C([H])=C12)=O)OC([H])([H])C1([H])C([H])([H])C1([H])[H])(=O)=O
Purity>98%
StoragePlease store the product under the recommended conditions in the Certificate of Analysis.

Biological Activity

CC-90010 (compound 1) is a reversible and orally active BET inhibitor. CC-90010 is applied in the study for advanced solid tumors

In Vitro

No in vitro data are provided in the current product source. Contact us for further information.

In Vivo

No in vivo data are provided in the current product source. Contact us for further information.

References & source

DC Chemicals original product information

Published experimental findings depend on the model and assay conditions. They do not guarantee equivalent performance in every application. For laboratory research use only.

Product documentation

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Handling guide

Please store the product under the recommended conditions in the Certificate of Analysis.

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