Denifanstat (TVB-2640) chemical structure
Chemical structureResearch use only
CAT. NO. DC26189Featured

Denifanstat (TVB-2640)

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TotalUS$950
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Product overview

Description & Application

TVB-2640(FASN-IN-2) is a Fatty Acid Synthase (FASN) inhibitor extracted from patent WO2012122391A1, compound 152, has an IC50 of 0.052 μM and an EC50 of 0.072 μM[1].

ParameterValue
Chemical Name4-(1-(4-Cyclobutyl-2-methyl-5-(5-methyl-4H-1,2,4-triazol-3- yl)benzoyl)piperidin-4-yl)benzonitrile
CAS No.1399177-37-7
SynonymsTVB-2640,TVB 2640,TVB2640
FormulaC27H29N5O
M.Wt439.55
SMILESC(C1C=CC(C2CCN(C(C3C(C)=CC(C4CCC4)=C(C4=NN=C(C)N4)C=3)=O)CC2)=CC=1)#N
Purity>98%
Storage2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO

Biological Activity

TVB-2640(FASN-IN-2) is a Fatty Acid Synthase (FASN) inhibitor extracted from patent WO2012122391A1, compound 152, has an IC50 of 0.052 μM and an EC50 of 0.072 μM[1].

In Vitro

No in vitro data are provided in the current product source. Contact us for further information.

In Vivo

No in vivo data are provided in the current product source. Contact us for further information.

References & source

DC Chemicals original product information

Published experimental findings depend on the model and assay conditions. They do not guarantee equivalent performance in every application. For laboratory research use only.

Product documentation

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Handling guide

2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO

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