RU-TRAAK-2 chemical structure
Chemical structureResearch use only
CAT. NO. DC22948Featured

RU-TRAAK-2

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TotalUS$800
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Product overview

Description & Application

RU-TRAAK-2 is a completely reversible TRAAK inhibitor, shows no activity for non-K2P channels (Kv1.2, Slo1 and GIRK2).

ParameterValue
Chemical Name1-(benzo[d]thiazol-2-ylmethyl)-1-methyl-3-(3-phenylprop-2-yn-1-yl)urea
CAS No.1210538-56-9
FormulaC19H17N3OS
M.Wt335.42
SMILESO=C(NCC#CC1=CC=CC=C1)N(CC2=NC3=CC=CC=C3S2)C
Purity>98%
Storage2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Biological Activity

RU-TRAAK-2 is a completely reversible TRAAK inhibitor, shows no activity for non-K2P channels (Kv1.2, Slo1 and GIRK2).

In Vitro

No in vitro data are provided in the current product source. Contact us for further information.

In Vivo

No in vivo data are provided in the current product source. Contact us for further information.

References & source

References 1. Su Z, et al. Proc Natl Acad Sci U S A. 2016 May 17;113(20):5748-53. 2. Cancer Res. 2017 Aug 15;77(16):4293-4304. View Related Products by Target Potassium Channel

DC Chemicals original product information

Published experimental findings depend on the model and assay conditions. They do not guarantee equivalent performance in every application. For laboratory research use only.

Product documentation

View online datasheetRequest COA / MSDS

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Handling guide

2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

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