GSK1016790A chemical structure
Chemical structureResearch use only
CAT. NO. DC11280Featured

GSK1016790A

Pack Sizes & Prices

TotalUS$800
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Product overview

Description & Application

GSK1016790A is a potent transient receptor potential vanilloid 4 (TRPV4) activator.

ParameterValue
Chemical Name(N-((1S)-1-{[4-((2S)-2-{[(2,4-Dichlorophenyl)sulfonyl]amino}-3-hydroxypropanoyl)-1-piperazinyl]carbonyl}-3-methylbutyl)-1-benzothiophene-2-carboxamide
CAS No.942206-85-1
SynonymsGSK1016790A,GSK-1016790A,GSK 1016790A
FormulaC28H32Cl2N4O6S2
M.Wt655.61
SMILESCC(C)C[C@@H](C(=O)N1CCN(CC1)C(=O)[C@H](CO)NS(=O)(=O)C2=C(C=C(C=C2)Cl)Cl)NC(=O)C3=CC4=CC=CC=C4S3
Purity>98%
Storage2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Biological Activity

GSK1016790A is a potent transient receptor potential vanilloid 4 (TRPV4) activator.

In Vitro

No in vitro data are provided in the current product source. Contact us for further information.

In Vivo

No in vivo data are provided in the current product source. Contact us for further information.

References & source

DC Chemicals original product information

Published experimental findings depend on the model and assay conditions. They do not guarantee equivalent performance in every application. For laboratory research use only.

Product documentation

View online datasheetRequest COA / MSDS

Refer to the certificate supplied with your lot for batch-specific release results.

Handling guide

2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Solution calculator

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