DSF-102 chemical structure
Chemical structureResearch use only
CAT. NO. DC74394Featured

DSF-102

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TotalUS$900
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Product overview

Description & Application

DSF-102 (DSF102) is a small molecule EGFR inhibitor that interacts with the extracellular domain (ECD) of EGFR, inhibits the interaction with the EGF instead of blocking the intracellular kinase activity, shows inhibition of EGFR dimerization with IC50 of

ParameterValue
Chemical Name2H-Indol-2-one, 1,3-dihydro-5-nitro-3-[[3-(trifluoromethyl)phenyl]imino]-
CAS No.197585-01-6
Synonyms2H-Indol-2-one, 1,3-dihydro-5-nitro-3-[[3-(trifluoromethyl)phenyl]imino]-
FormulaC15H8N3O3F3
M.Wt335.238
SMILES[N+](C1C=CC2=C(/C(=N/C3C=CC=C(C(F)(F)F)C=3)/C(=O)N2)C=1)([O-])=O
Purity>98%
Storage2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Biological Activity

DSF-102 (DSF102) is a small molecule EGFR inhibitor that interacts with the extracellular domain (ECD) of EGFR, inhibits the interaction with the EGF instead of blocking the intracellular kinase activity, shows inhibition of EGFR dimerization with IC50 of

In Vitro

No in vitro data are provided in the current product source. Contact us for further information.

In Vivo

No in vivo data are provided in the current product source. Contact us for further information.

References & source

DC Chemicals original product information

Published experimental findings depend on the model and assay conditions. They do not guarantee equivalent performance in every application. For laboratory research use only.

Product documentation

View online datasheetRequest COA / MSDS

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Handling guide

2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Solution calculator

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