DP308 chemical structure
Chemical structureResearch use only
CAT. NO. DC73322Featured

DP308

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TotalUS$450
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Product overview

Description & Application

DP308 is a novel and effective 53BP1 tandem Tudor domain (TTD) inhibitor, disrupts the binding between 53BP1 and H4K20me2 peptide with IC50 of 1.69 uM.

ParameterValue
Chemical NameDP308
CAS No.685884-37-1
SynonymsDP-308;DP 308
FormulaC21H23N3O2
M.Wt349.43
SMILESCCN(CC)C1=CC(C)=C2C=C(NC(=O)/C=C/C3=CC=CO3)C=CC2=N1
Purity>98%
Storage2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Biological Activity

DP308 is a novel and effective 53BP1 tandem Tudor domain (TTD) inhibitor, disrupts the binding between 53BP1 and H4K20me2 peptide with IC50 of 1.69 uM.

In Vitro

No in vitro data are provided in the current product source. Contact us for further information.

In Vivo

No in vivo data are provided in the current product source. Contact us for further information.

References & source

DC Chemicals original product information

Published experimental findings depend on the model and assay conditions. They do not guarantee equivalent performance in every application. For laboratory research use only.

Product documentation

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Handling guide

2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

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