DC Chemicals · Product datasheet

Ver-246608 — Datasheet

CAT. NO. DCC5399

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ParameterValue
Chemical NameVER-246608
CAS No.1684386-71-7
SynonymsN-[4-(2-Chloro-5-Methylpyrimidin-4-Yl)phenyl]-N-(4-{[(Difluoroacetyl)amino]methyl}benzyl)-2,4-Dihydroxybenzamide;N-[4-(2-chloro-5-methylpyrimidin-4-yl)phenyl]-N-[[4-[[(2,2-difluoroacetyl)amino]methyl]phenyl]methyl]-2,4-dihydroxybenzamide;N-(4-(2-chloro-5-methylpyrimidin-4-yl)phenyl)-N-(4-((2,2-difluoroacetamido)methyl)benzyl)-2,4-dihydroxybenzamide;N-[4-(2-Chloro-5-methyl-4-pyrimidinyl)phenyl]-N-[[4-[[(2,2-difluoroacetyl)amino]methyl]phenyl]methyl]-2,4-dihyd;VER-246608;N-[4-(2-chloro-5-methylpyrimidin-4-yl)phenyl]-N-({4-[(2,2-difluoroacetamido)methyl]phenyl}methyl)-2,4-dihydroxybenzamide;N-[4-(2-chloro-5-methylpyrimidin-4-yl)phenyl]-N-({4-[(2,2-difluoroacetamido)methyl]phenyl}methyl)-2,4-dihydroxybenzamide;N-(4-(2-chloro-5-methylpyrimidin-4-yl)phenyl)-N-((4-(((2,2-difluoroacetyl)amino)methyl)phenyl)methyl)-2,4-dihydroxybenzamide;N-(4-(2-chloro-5-methylpyrimidin-4-yl)phenyl)-N-((4-(((2,2-difluoroacetyl)amino)methyl)phenyl)methyl)-2,4-dihydroxybenzamide;MS-30103;MS-30103;SZ6;SZ6;AKOS040742812;AKOS040742812;N-[4-(2-Chloro-5-methyl-4-pyrimidinyl)phenyl]-N-[[4-[[(2,2-difluoroacetyl)amino]methyl]phenyl]methyl]-2,4-dihydroxy-benzamide;N-[4-(2-Chloro-5-methyl-4-pyrimidinyl)phenyl]-N-[[4-[[(2,2-difluoroacetyl)amino]methyl]phenyl]methyl]-2,4-dihydroxy-benzamide;1684386-71-7;1684386-71-7;CHEMBL3727577;CHEMBL3727577;VER 246608; VER246608;VER 246608; VER246608;DA-58983;DA-58983;CS-0011787;CS-0011787;SCHEMBL16586236;SCHEMBL16586236;G14475;G14475;Q27465596;Q27465596;GTPL9350;GTPL9350;4v25;4v25;EX-A3785;EX-A3785;LCGNLQSOSJFLKR-UHFFFAOYSA-N;LCGNLQSOSJFLKR-UHFFFAOYSA-N;BDBM50236530;BDBM50236530;BCP29722;BCP29722;HY-12492;HY-12492
FormulaC28H23ClF2N4O4
M.Wt552.956432580948
SMILESClC1=NC=C(C)C(C2C=CC(=CC=2)N(C(C2C=CC(=CC=2O)O)=O)CC2C=CC(CNC(C(F)F)=O)=CC=2)=N1
Purity98%
Storage2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Biological Activity

Novel pan-isoform ATP competitive inhibitor of pyruvate dehydrogenase kinase, disrupting Warburg metabolism and inducing context-dependent cytostasis in cancer cells

In Vitro

No in vitro data are provided in the current product source. Contact us for further information.

In Vivo

No in vivo data are provided in the current product source. Contact us for further information.

References & source

DC Chemicals original product information

Published experimental findings depend on the model and assay conditions. They do not guarantee equivalent performance in every application. For laboratory research use only.

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