AP-III-a4 hydrochloride Datasheet | DC9247

AP-III-a4 hydrochloride — Datasheet

CAT. NO. DC9247

Parameter	Value
Chemical Name	AP-III-a4 hydrochloride
CAS No.	2070014-95-6
Synonyms	Benzeneacetamide, N-[2-[2-(2-aminoethoxy)ethoxy]ethyl]-4-[[4-[(cyclohexylmethyl)amino]-6-[[(4-fluorophenyl)methyl]amino]-1,3,5-triazin-2-yl]amino]-, hydrochloride;AP-III-a4 hydrochloride
Formula	C31H44ClFN8O3
M.Wt	631.18
SMILES	C1CCC(CNC2=NC(=NC(NC3=CC=C(C=C3)CC(NCCOCCOCCN)=O)=N2)NCC2C=CC(F)=CC=2)CC1.Cl
Purity	>98%
Storage	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Biological Activity

ENOblock Hcl(AP-III-a4 Hcl) is a novel small molecule which is the first, nonsubstrate analogue that directly binds to enolase and inhibits its activity (IC50=0.576 uM); inhibit cancer cell metastasis in vivo.

In Vitro

No in vitro data are provided in the current product source. Contact us for further information.

In Vivo

No in vivo data are provided in the current product source. Contact us for further information.

References & source

DC Chemicals original product information

Published experimental findings depend on the model and assay conditions. They do not guarantee equivalent performance in every application. For laboratory research use only.

AP-III-a4 hydrochloride — Datasheet

Biological Activity

In Vitro

In Vivo

References & source

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