DC Chemicals · Product datasheet

TAS-116 — Datasheet

CAT. NO. DC8142

Product page and current package options

ParameterValue
Chemical NamePimitespib
CAS No.1260533-36-5
SynonymsPLO044MUDZ;Pimitespib;Tas 116;TAS116 pound>>TAS 116;BDBM126083;BCP25132;NSC780204;s7716;DB14876;SB17223;US8779142, 102;3-Ethyl-4-(3-(1-methylethyl)-4-(4-(1-methyl-1H-pyrazol-4-yl)-1H-imidazol-1-yl)-1H-pyrazolo(3,4-b)pyridin-1-yl)benzamide;3-ethyl-4-(3-isopropyl-4-(4-(1-methyl-1H-pyrazol-4-yl)-1H-imidazol-1-yl)-1H-pyrazolo[3,4-b]pyridin-1-yl)benzamide;3-ethyl-4-[;Tas-116;TAS 116，TAS116
FormulaC25H26N8O
M.Wt454.526943683624
SMILESO=C(C1C=CC(=C(C=1)CC)N1C2C(=C(C=CN=2)N2C=NC(C3C=NN(C)C=3)=C2)C(C(C)C)=N1)N
Purity>96%
Storage2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO

Biological Activity

TAS-116 is a potent and selective HSP90α/β inhibitor with Kis of 34.7 nM, 21.3 nM, respectively.

In Vitro

No in vitro data are provided in the current product source. Contact us for further information.

In Vivo

No in vivo data are provided in the current product source. Contact us for further information.

References & source

DC Chemicals original product information

Published experimental findings depend on the model and assay conditions. They do not guarantee equivalent performance in every application. For laboratory research use only.

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