DC Chemicals · Product datasheet

MS8815 — Datasheet

CAT. NO. DC72540

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ParameterValue
Chemical NameMS8815
CAS No.2855085-25-3
SynonymsMS8815;MS 8815
FormulaC65H87N9O8S
M.Wt1154.50679516792
SMILESN(C1CCOCC1)(C1C(C)=C(C(=O)NCC2C(=O)NC(C)=CC=2C)C=C(C2C=CC(CN3CCN(C(=O)CCCCCCCC(=O)N[C@@H](C(C)(C)C)C(N4C[C@H](O)C[C@H]4C(=O)NCC4C=CC(C5SC=NC=5C)=CC=4)=O)CC3)=CC=2)C=1)CC
Purity98%
Storage2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Biological Activity

MS8815 is a selective enhancer of zeste homolog 2 (EZH2) PROTAC degrader. MS8815 has inhibition activity for EZH2 with an IC50 value of 8.6 nM. MS8815 can be used for the research of triple-negative breast cancer (TNBC).

In Vitro

No in vitro data are provided in the current product source. Contact us for further information.

In Vivo

No in vivo data are provided in the current product source. Contact us for further information.

References & source

DC Chemicals original product information

Published experimental findings depend on the model and assay conditions. They do not guarantee equivalent performance in every application. For laboratory research use only.

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