DC Chemicals · Product datasheet

Emraclidine — Datasheet

CAT. NO. DC46844

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Parameter	Value
Chemical Name	Unii-J241Y80eeo
CAS No.	2170722-84-4
Synonyms	J241Y80EEO;Emraclidine;Emraclidine [INN];1-(2,4-Dimethyl-5,7-dihydro-6H-pyrrolo(3,4-b)pyridin-6-yl)-2-(1-(2-(trifluoromethyl)pyridin-4-yl)azetidin-3-yl)ethan-1-one;Ethanone, 1-(5,7-dihydro-2,4-dimethyl-6H-pyrrolo(3,4-b)pyridin-6-yl)-2-(1-(2-(trifluoromethyl)-4-pyridinyl)-3-azetidinyl)-;Unii-J241Y80eeo
Formula	C20H21F3N4O
M.Wt	390.4022
SMILES	FC(C1C([H])=C(C([H])=C([H])N=1)N1C([H])([H])C([H])(C([H])([H])C(N2C([H])([H])C3=C(C(C([H])([H])[H])=C([H])C(C([H])([H])[H])=N3)C2([H])[H])=O)C1([H])[H])(F)F
Purity	>98%
Storage	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Biological Activity

Emraclidine is a muscarinic M4 receptor positive allosteric modulator (WO2018002760, compound 11). Emraclidine can be used for the research of neurological diseases.

In Vitro

Emraclidine is a muscarinic M4 receptor positive allosteric modulator[1].

In Vivo

No in vivo data are provided in the current product source. Contact us for further information.

Target

Muscarinic M4 Receptor[1]

References & source

[1]. WO2018002760

DC Chemicals original product information

Published experimental findings depend on the model and assay conditions. They do not guarantee equivalent performance in every application. For laboratory research use only.