DC Chemicals · Product datasheet

J-2156 TFA — Datasheet

CAT. NO. DC44000

Product page and current package options

ParameterValue
Chemical NameJ-2156 TFA
CAS No.2387505-73-7
SynonymsJ-2156 TFA;Unk-Dab-Phe-NH2.TFA;J-2156 (TFA);(S)-4-AMino-N-((S)-1-amino-1-oxo-3-phenylpropan-2-yl)-2-((4-methylnaphthalene)-1-sulfonamido)butanamide 2,2,2-trifluoroacetate;2387505-73-7;HY-111615A;(2S)-4-amino-N-[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]-2-[(4-methylnaphthalen-1-yl)sulfonylamino]butanamide;2,2,2-trifluoroacetic acid;MS-30439;CS-0120693;G17691
FormulaC26H29F3N4O6S
M.Wt582.59187579155
SMILESS(C1=CC=C(C)C2C=CC=CC1=2)(N[C@H](C(N[C@H](C(N)=O)CC1C=CC=CC=1)=O)CCN)(=O)=O.FC(C(=O)O)(F)F
Purity>98%
Storage2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Biological Activity

J-2156 TFA is a high potent, selective somatostatin receptor type 4 (SST4 receptor) agonist with IC50s of 0.05 nM and 0.07 nM for human and rat SST4 receptors, respectively. J-2156 TFA is used for the relief of mechanical allodynia and mechanical hyperalg

In Vitro

No in vitro data are provided in the current product source. Contact us for further information.

In Vivo

No in vivo data are provided in the current product source. Contact us for further information.

References & source

DC Chemicals original product information

Published experimental findings depend on the model and assay conditions. They do not guarantee equivalent performance in every application. For laboratory research use only.

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