DC Chemicals · Product datasheet

ERAP1-IN-1 — Datasheet

CAT. NO. DC28740

Product page and current package options

ParameterValue
Chemical NameErap1-IN-1
CAS No.865273-97-8
SynonymsERAP1-IN-1;MLS002163123;KUC114049N;KUC114390N;SMR001245516;Z45705491;4-methoxy-3-{[2-(piperidin-1-yl)-5-(trifluoromethyl)phenyl]sulfamoyl}benzoic acid;4-Methoxy-3-[[[2-(1-piperidinyl)-5-(trifluoromethyl)phenyl]amino]sulfonyl]benzoic acid (ACI);4-Methoxy-3-(N-(2-(piperidin-1-yl)-5-(trifluoromethyl)phenyl)sulfamoyl)benzoic Acid;4-Methoxy-3-[N-[2-(piperidin-1-yl)-5-(trifluoromethyl)phenyl]sulfamoyl]benzoic acid
FormulaC20H21F3N2O5S
M.Wt458.45135474205
SMILESO=C(C1C=C(S(NC2C(N3CCCCC3)=CC=C(C(F)(F)F)C=2)(=O)=O)C(OC)=CC=1)O
Purity>98%
Storage2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Biological Activity

ERAP1-IN-1 is an endoplasmic reticulum aminopeptidase 1 (ERAP1) inhibitor. ERAP1-IN-1 competitively inhibits ERAP1 activity towards a nonamer peptide representative of physiological substrates.

In Vitro

No in vitro data are provided in the current product source. Contact us for further information.

In Vivo

No in vivo data are provided in the current product source. Contact us for further information.

References & source

DC Chemicals original product information

Published experimental findings depend on the model and assay conditions. They do not guarantee equivalent performance in every application. For laboratory research use only.

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