DC Chemicals · Product datasheet

GR-127935 hydrochloride — Datasheet

CAT. NO. DC21064

Product page and current package options

ParameterValue
Chemical NameN-[4-methoxy-3-(4-methylpiperazin-1-yl)phenyl]-4-[2-methyl-4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]benzamide hydrochloride
CAS No.148642-42-6
SynonymsGR127935
FormulaC29H31N5O3.HCl
M.Wt534.06
SMILESCl.CN1CCN(C2C=C(NC(C3C=CC(C4C=CC(C5=NOC(C)=N5)=CC=4C)=CC=3)=O)C=CC=2OC)CC1
Purity>98%
Storage2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Biological Activity

GR-127935 potent and selective 5-HT1B/1D receptor antagonist with pKi of 8.5 for both guinea pig 5-HT1D and rat 5-HT1B receptor.

In Vitro

No in vitro data are provided in the current product source. Contact us for further information.

In Vivo

No in vivo data are provided in the current product source. Contact us for further information.

References & source

DC Chemicals original product information

Published experimental findings depend on the model and assay conditions. They do not guarantee equivalent performance in every application. For laboratory research use only.

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