DC Chemicals · Product datasheet

HC-067047 — Datasheet

CAT. NO. DC11416

Product page and current package options

ParameterValue
Chemical Name2-Methyl-1-(3-morpholin-4-ylpropyl)-5-phenyl-N-[3-(trifluoromethyl)phenyl]pyrrole-3-carboxamide
CAS No.883031-03-6
SynonymsHC 067047;HC-067047;2-methyl-1-(3-morpholin-4-ylpropyl)-5-phenyl-N-[3-(trifluoromethyl)phenyl]pyrrole-3-carboxamide;2-Methyl-1-[3-(4-morpholinyl)propyl]-5-phenyl-N-[3-(trifluoromethyl)phenyl]-1H-pyrrole-3-carboxamide;HC067047;MLS006012019;GTPL4213;AOB5050;ONC 212;HMS3743C07;BCP34020;BDBM50192821;s6637;SMR0047035
FormulaC26H28F3N3O2
M.Wt471.5146
SMILESFC(C1C([H])=C([H])C([H])=C(C=1[H])N([H])C(C1C([H])=C(C2C([H])=C([H])C([H])=C([H])C=2[H])N(C=1C([H])([H])[H])C([H])([H])C([H])([H])C([H])([H])N1C([H])([H])C([H])([H])OC([H])([H])C1([H])[H])=O)(F)F
Purity>98%
Storage2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Biological Activity

HC-067047 is a potent and selective TRPV4 antagonist with IC50s of 48 nM, 133 nM, and 17 nM for human, rat, and mouse TRPV4.

In Vitro

No in vitro data are provided in the current product source. Contact us for further information.

In Vivo

No in vivo data are provided in the current product source. Contact us for further information.

References & source

DC Chemicals original product information

Published experimental findings depend on the model and assay conditions. They do not guarantee equivalent performance in every application. For laboratory research use only.

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