p38-α MAPK-IN-1 Datasheet | DC10798

p38-α MAPK-IN-1 — Datasheet

CAT. NO. DC10798

Parameter	Value
Chemical Name	MAPK14 inhibitor
CAS No.	443913-15-3
Synonyms	MAPK14 inhibitor
Formula	C27H35N5O3
M.Wt	477.6
SMILES	CC1=CC=C(N2C(NC(NC3=CC=C(OCCN4CCOCC4)C=C3)=O)=CC(C(C)(C)C)=N2)C=C1
Purity	>98%
Storage	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Biological Activity

p38-α MAPK-IN-1 is an inhibitor of MAPK14 (p38-α), with IC50 of 2300 nM in EFC displacement assay, and 5500 nM in HTRF assay.

In Vitro

p38-α MAPK-IN-1 (Compound 12) is an inhibitor of MAPK14 (p38-α)>, with IC50 of 2300 nM in EFC displacement assay, and 5500 nM in HTRF assay[1].

In Vivo

No in vivo data are provided in the current product source. Contact us for further information.

References & source

DC Chemicals original product information

Published experimental findings depend on the model and assay conditions. They do not guarantee equivalent performance in every application. For laboratory research use only.

p38-α MAPK-IN-1 — Datasheet

Biological Activity

In Vitro

In Vivo

References & source

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